Compile Data Set for Download or QSAR
maximum 50k data
Found 101 of ki data for polymerid = 49000381,49000382,50000031,50006274
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50055978(4-((R)-2-Cyclohexyl-2-hydroxy-2-phenyl-acetoxy)-1,...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M3 was determined in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50055976((R)-3-((R)-2-Cyclohexyl-2-hydroxy-2-phenyl-acetoxy...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M3 was determined in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82372(CAS_22254-24-6 | Ipratropium | NSC_3746)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM50015720((hyoscine)3-Hydroxy-2-phenyl-propionic acid 9-meth...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50015720((hyoscine)3-Hydroxy-2-phenyl-propionic acid 9-meth...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50010096(CHEMBL12980 | Hydroxy-diphenyl-acetic acid 1-aza-b...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50151858(4-(diethylamino)but-2-yn-1-yl (2S)-cyclohexyl(hydr...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM81800(CAS_57558-44-8 | NSC_42470 | Secoverine)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50369230(CHEMBL1398637 | CLIDINIUM)
Affinity DataKi:  0.650nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M3 was determined in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM86698(BENZTROPINE | CAS_132-17-2 | CHEMBL116590 | NSC_23...)
Affinity DataKi:  0.890nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM82423(CAS_132947 | NSC_132947 | TRIPITRAMINE)
Affinity DataKi:  0.970nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82379(BTM 1042 hydrochloride | BTM1086 | CAS_87687-13-6)
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)
Affinity DataKi:  1.41nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50010101(2-(diethylamino)ethyl 1-cyclohexylcyclohexanecarbo...)
Affinity DataKi:  1.51nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM81462((R)-Trihexyphenidyl | (S)-Trihexyphenidyl | Benzhe...)
Affinity DataKi:  1.95nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)
Affinity DataKi:  2.04nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50240680(1-(bicyclo[2.2.1]hept-5-en-2-yl)-1-phenyl-3-(piper...)
Affinity DataKi:  2.04nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82375(CAS_512-15-2 | Cyclopentolate | NSC_2905)
Affinity DataKi:  2.57nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  2.63nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50005685(2,2-Diphenyl-propionic acid 2-diethylamino-ethyl e...)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50010096(CHEMBL12980 | Hydroxy-diphenyl-acetic acid 1-aza-b...)
Affinity DataKi:  4.60nMAssay Description:In vitro binding affinity against against guinea pig ileum using [3H]-N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50062598(1-Cyclohexyl-1-phenyl-3-pyrrolidin-1-yl-propan-1-o...)
Affinity DataKi:  4.79nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82374(Botiacrine | CAS_4774-53-2 | NSC_71202)
Affinity DataKi:  5.13nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82380(CAS_36167-80-3 | PrBCh | Propylbenzilylcholine Mus...)
Affinity DataKi:  5.89nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  6.17nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50034874((R)-Hydroxy-(4-iodo-phenyl)-phenyl-acetic acid 1-a...)
Affinity DataKi:  8.10nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]-N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM50071173((3R,4R,4aS,8aR)-4-[(E)-2-((2S,6S)-1,6-Dimethyl-pip...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM82376(CAS_80880-90-6 | NSC_5387 | TELENZEPINE)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82371(CAS_1508-75-4 | NSC_5593 | TROPICAMIDE)
Affinity DataKi:  14.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  15.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82373(DABDMA | diphenylacetoxybutynyl dimethylamine)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82370(CAS_87-00-3 | Homatropine | NSC_5821)
Affinity DataKi:  25.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  32.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  33.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  34.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50034873((S)-(4-Fluoromethyl-phenyl)-hydroxy-phenyl-acetic ...)
Affinity DataKi:  39nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]-N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50034873((S)-(4-Fluoromethyl-phenyl)-hydroxy-phenyl-acetic ...)
Affinity DataKi:  39nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]-N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50034870((S)-Hydroxy-(4-iodo-phenyl)-phenyl-acetic acid 1-a...)
Affinity DataKi:  41nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]-N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM82371(CAS_1508-75-4 | NSC_5593 | TROPICAMIDE)
Affinity DataKi:  41.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  55.0nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50034872((S)-[4-(3-Fluoro-propyl)-phenyl]-hydroxy-phenyl-ac...)
Affinity DataKi:  59nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]-N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50036185(3-(2'-Benzofuranyl)-quinuclidine-2-ene | 3-Benzofu...)
Affinity DataKi:  59nMAssay Description:Binding affinity for muscarinic acetylcholine receptor M3 by measuring displacement of [3H]-QNB from guinea pig parotid glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM82378(CAS_82-98-4 | NSC_4839 | Piperidolate)
Affinity DataKi:  64.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)
Affinity DataKi:  67nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M3 was determined in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(PORCINE)
Case Western Reserve University

Curated by PDSP Ki Database
LigandPNGBDBM85381(CAS_116679-83-5 | p-FHSD | p-fluoro-hexahydro-sila...)
Affinity DataKi:  69.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50407330(CHEMBL2112939)
Affinity DataKi:  80nMAssay Description:In vitro binding affinity towards Muscarinic acetylcholine receptor M3 was determined by measuring its ability to displace [3H]-N-methyl- scopolamine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(RABBIT)
Glaxo Group Research

Curated by PDSP Ki Database
LigandPNGBDBM50062614(CHEMBL900 | Dimethyl-[2-(phenyl-o-tolyl-methoxy)-e...)
Affinity DataKi:  81.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Groningen University Hospital

Curated by ChEMBL
LigandPNGBDBM50034875((S)-[4-(2-Fluoro-ethyl)-phenyl]-hydroxy-phenyl-ace...)
Affinity DataKi:  85nMAssay Description:In vitro binding affinity against guinea pig ileum using [3H]-N-methylscopolamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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